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Targets Recommended: p38 MAPK

3

抑制剂 & 化合物

4

天然产物

4

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T11943 MAPK13-IN-1

p38 MAPK MAPK
MAPK13-IN-1 是一种有效的 MAPK13 (p38δ) 抑制剂(IC50:620 nM)。
T3462 BMS-582949 hydrochloride

BMS-582949 HCl

p38 MAPK; Autophagy Autophagy; MAPK
BMS-582949 hydrochloride (BMS-582949 HCl) 是一种高度特异性的 p38α MAPK 抑制剂,其 IC50值为13 nM,可研究炎症性疾病。
T6789 BMS582949

BMS 582949,PS540446,BMS-582949

p38 MAPK MAPK
BMS582949 (PS540446) 是一种有效的选择性 p38 丝裂原活化蛋白激酶(p38 MAPK) 抑制剂,IC50 为 13 nM,抑制 p38 激酶活性和 p38 活化。

化合物

MAPK13-IN-1
Cat.No: T11943
Synonym:
Target: p38 MAPK
BMS-582949 hydrochloride
Cat.No: T3462
Synonym: BMS-582949 HCl
Target: p38 MAPK, Autophagy
BMS582949
Cat.No: T6789
Synonym: BMS 582949,PS540446,BMS-582949
Target: p38 MAPK
Cat. No. Product Name Target Signaling Pathways
T5S2358 Dehydrocorydaline

Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T10990 Dehydrocorydaline chloride

盐酸脱氢紫堇碱,13-Methylpalmatine chloride

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T9218 Andrograpanin

19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE,新穿心莲内酯苷元

p38 MAPK MAPK
Andrograpanin (19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE) 是来自穿心莲的一种天然产物,具有抗炎和抗感染活性。
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。

天然产物

Dehydrocorydaline
Cat.No: T5S2358
Synonym: Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Dehydrocorydaline chloride
Cat.No: T10990
Synonym: 盐酸脱氢紫堇碱,13-Methylpalmatine chloride
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Andrograpanin
Cat.No: T9218
Synonym: 19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE,新穿心莲内酯苷元
Target: p38 MAPK
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Cat. No. Product Name Species Expression System
TMPY-04551 p38 delta/MAPK13 Protein, Human, Recombinant (GST)

MAPK13,p38δ,PRKM13,MAPK-...

Human Baculovirus Insect Cells
p38 delta/MAPK13 Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 68.4 kDa and the accession number is O15264.
TMPY-04531 p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro

P38 δ/MAPK13,MAPK13,PRKM...

Human Baculovirus Insect Cells
p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 68.4 kDa and the accession number is O15264.
TMPK-01373 Fibronectin Protein, Human, Recombinant (aa 1266-1356, hFc)

FINC,LETS,GFND,SMDCF,GFND2,ED-B,MSF,FNZ,FN1,FN,CIG

Human HEK293 Cells
Fibronectin is a high molecular glycoprotein present in the blood, connective tissue and at cell surface. It is synthesized by many types of differentiated cells and is believed to be involved in the attachment of cells to the surrounding extracellular matrix. Fibronectin has affinity to the other main components of extracellular matrix, collagen and glycosaminoglycans. Fibronectin Protein, Human, Recombinant (aa 1266-1356, hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicte...
TMPK-01391 Fibronectin Protein, Human, Recombinant (aa 1266-1356, His)

FN1,LETS,GFND,MSF,FNZ,CIG,ED-B,FN,SMDCF,GFND2,FINC

Human HEK293 Cells
Fibronectin is a high molecular glycoprotein present in the blood, connective tissue and at cell surface. It is synthesized by many types of differentiated cells and is believed to be involved in the attachment of cells to the surrounding extracellular matrix. Fibronectin has affinity to the other main components of extracellular matrix, collagen and glycosaminoglycans. Fibronectin Protein, Human, Recombinant (aa 1266-1356, His) is expressed in HEK293 mammalian cells with C-His tag. The predicte...

重组蛋白

p38 delta/MAPK13 Protein, Human, Recombinant (GST)
Cat.No: TMPY-04551
Species: Human
Expression System: Baculovirus Insect Cells
p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro
Cat.No: TMPY-04531
Species: Human
Expression System: Baculovirus Insect Cells
Fibronectin Protein, Human, Recombinant (aa 1266-1356, hFc)
Cat.No: TMPK-01373
Species: Human
Expression System: HEK293 Cells
Fibronectin Protein, Human, Recombinant (aa 1266-1356, His)
Cat.No: TMPK-01391
Species: Human
Expression System: HEK293 Cells
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